发明名称 |
Composition for treating or preventing glaucoma comprising a sulfonamide compound, and a beta-receptor antagonist |
摘要 |
A composition for treating or preventing glaucoma or ocular hypertension including a isopropyl (6-{[4-(pyrazol-1-yl)benzyl](pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino)acetate and a beta-receptor antagonist, in a combined pharmaceutically acceptable amount. As for the administration form, these drugs may be administered concomitantly or may be administered as a combination drug. |
申请公布号 |
US9339496(B2) |
申请公布日期 |
2016.05.17 |
申请号 |
US201313939381 |
申请日期 |
2013.07.11 |
申请人 |
SANTEN PHARMACEUTICAL CO., LTD. |
发明人 |
Kirihara Tomoko;Shimazaki Atsushi;Nakamura Masatsugu |
分类号 |
A61K31/444;A61K45/06;C07D401/14;A61K31/498;A61K31/5377;A61K31/542;A61K31/5575 |
主分类号 |
A61K31/444 |
代理机构 |
Holtz, Holtz & Volek PC |
代理人 |
Holtz, Holtz & Volek PC |
主权项 |
1. A composition for treating glaucoma or ocular hypertension comprising 0.001 to 0.1 w/v % of isopropyl (6-{[4-(pyrazol-1-yl)benzyl](pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino)acetate and 0.1 to 0.5 w/v % of timolol, in a combined pharmaceutically effective amount, wherein the isopropyl (6-{[4-(pyrazol-1-yl)benzyl](pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino)acetate may be in the form of a salt thereof, and the timolol may be in the form of a salt thereof. |
地址 |
Osaka JP |