发明名称 Composition for treating or preventing glaucoma comprising a sulfonamide compound, and a beta-receptor antagonist
摘要 A composition for treating or preventing glaucoma or ocular hypertension including a isopropyl (6-{[4-(pyrazol-1-yl)benzyl](pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino)acetate and a beta-receptor antagonist, in a combined pharmaceutically acceptable amount. As for the administration form, these drugs may be administered concomitantly or may be administered as a combination drug.
申请公布号 US9339496(B2) 申请公布日期 2016.05.17
申请号 US201313939381 申请日期 2013.07.11
申请人 SANTEN PHARMACEUTICAL CO., LTD. 发明人 Kirihara Tomoko;Shimazaki Atsushi;Nakamura Masatsugu
分类号 A61K31/444;A61K45/06;C07D401/14;A61K31/498;A61K31/5377;A61K31/542;A61K31/5575 主分类号 A61K31/444
代理机构 Holtz, Holtz & Volek PC 代理人 Holtz, Holtz & Volek PC
主权项 1. A composition for treating glaucoma or ocular hypertension comprising 0.001 to 0.1 w/v % of isopropyl (6-{[4-(pyrazol-1-yl)benzyl](pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino)acetate and 0.1 to 0.5 w/v % of timolol, in a combined pharmaceutically effective amount, wherein the isopropyl (6-{[4-(pyrazol-1-yl)benzyl](pyridin-3-ylsulfonyl)aminomethyl}pyridin-2-ylamino)acetate may be in the form of a salt thereof, and the timolol may be in the form of a salt thereof.
地址 Osaka JP