发明名称 Heterocyclic compounds as pesticides
摘要 The present application relates to novel amides and thioamides, to processes for preparation thereof and to the use thereof for controlling animal pests, in particular arthropods and especially insects.
申请公布号 US9339032(B2) 申请公布日期 2016.05.17
申请号 US201414156897 申请日期 2014.01.16
申请人 Bayer Intellectual Property GmbH 发明人 Bretschneider Thomas;Köhler Adeline;Fischer Reiner;Fublein Martin;Jeschke Peter;Kluth Joachim;Mühlthau Friedrich August;Voerste Arnd;Malsam Olga;Görgens Ulrich;Sato Yoshitaka
分类号 A01N43/56;A01N43/54;A01N43/40;A01N43/78;A01N47/02;C07D401/04;C07D417/04;C07D417/14 主分类号 A01N43/56
代理机构 Sterne, Kessler, Goldstein & Fox P.L.L.C. 代理人 Sterne, Kessler, Goldstein & Fox P.L.L.C.
主权项 1. A compound of formula (I), a salt thereof, or an N-oxide thereof, in which A1 and A2 are each independently hydrogen, halogen, cyano, nitro, alkyl, cycloalkyl or alkoxy, G1 is N or C-A1, and G2 is a radical selected from the group consisting of in which the arrow marks the bond to the adjacent ring, R1 in the case of the heterocycles (A) and (D) is hydrogen, halogen, cyano, alkyl, alkoxy, amino, alkylamino, dialkylamino, alkylthio or haloalkyl, or R1 in the case of heterocycle (C) is hydrogen, alkyl or haloalkyl, B is hydrogen, halogen, cyano, nitro, alkyl, cycloalkyl, haloalkyl, amino, alkylamino, dialkylamino, alkylthio or alkoxy, and G3 is a radical selected from the group consisting of in which the arrow marks the bond to G2 and the radicals (F), (G), (H), (K) and (L) can be combined with the heterocycles (A), (B), (C) and (D), and the radical (J) can be combined with the heterocycles (A), (C) and (D), X is oxygen or sulphur, n is 1 or 2, R2 is hydrogen, alkyl, haloalkyl, cyanoalkyl, alkoxy, haloalkoxy, alkenyl, alkoxyalkyl, optionally halogen-substituted alkylcarbonyl, optionally halogen-substituted alkoxycarbonyl, optionally halogen-, alkyl-, alkoxy-, haloalkyl- or cyano-substituted cycloalkylcarbonyl, or a cation, R3 and R7 are each independently in each case optionally substituted alkyl, alkenyl, or alkynyl, in each case optionally substituted cycloalkyl, cycloalkylalkyl, or cycloalkenyl, in which the rings optionally contain at least one heteroatom selected from the group consisting of sulphur, oxygen (where oxygen atoms must not be immediately adjacent) and nitrogen, in each case optionally substituted aryl, heteroaryl, arylalkyl or heteroarylalkyl, or an optionally substituted amino group, or R2 and R3 optionally form, together with the N—S(O)n group to which they are bonded, a saturated or unsaturated and optionally substituted 4- to 8-membered ring which optionally contain one or more further heteroatoms selected from the group consisting of sulphur, oxygen (where oxygen atoms must not be immediately adjacent) and nitrogen, and/or optionally contain at least one carbonyl group, R4 and R5 are each independently in each case optionally substituted alkyl, alkenyl, alkoxy, or alkynyl, in each case optionally substituted cycloalkyl, cycloalkylalkyl, or cycloalkenyl, in which the rings optionally contain at least one heteroatom selected from the group consisting of sulphur, oxygen (where oxygen atoms must not be immediately adjacent) and nitrogen, in each case optionally substituted aryl, heteroaryl, arylalkyl or heteroarylalkyl, or an optionally substituted amino group, R8 is hydrogen, optionally substituted alkyl, alkenyl, alkoxy, or alkynyl, optionally substituted cycloalkyl, cycloalkylalkyl, or cycloalkenyl, in which the rings optionally contain at least one heteroatom selected from the group consisting of sulphur, oxygen (where oxygen atoms must not be immediately adjacent) and nitrogen, optionally substituted aryl, heteroaryl, arylalkyl or heteroarylalkyl, or an optionally substituted amino group, R2 and R5 optionally form, together with the N—C(X) group to which they are bonded, a saturated or unsaturated and optionally substituted 4- to 8-membered ring which optionally contain one or more further heteroatoms selected from the group consisting of sulphur, oxygen (where oxygen atoms must not be immediately adjacent) and nitrogen, and/or optionally contain at least one carbonyl group, R6 is hydrogen or alkyl, R2 and R6 optionally form, together with the nitrogen atoms to which they are bonded, a saturated or unsaturated and optionally substituted 4- to 8-membered ring which optionally contain at least one further heteroatom selected from the group consisting of sulphur, oxygen (where oxygen atoms must not be immediately adjacent) and nitrogen, and/or optionally contain at least one carbonyl group, R6 and R7 optionally form, together with the N—S(O)n group to which they are bonded, a saturated or unsaturated and optionally substituted 4- to 8-membered ring which optionally contain one or more further heteroatoms selected from the group consisting of sulphur, oxygen (where oxygen atoms must not be immediately adjacent) and nitrogen, and/or optionally contain at least one carbonyl group, R2 and R8 optionally form, together with the nitrogen atom to which they are bonded, a saturated or unsaturated and optionally substituted 4- to 8-membered ring which optionally contain one or more further heteroatoms selected from the group consisting of sulphur, oxygen (where oxygen atoms must not be immediately adjacent) and nitrogen, and/or optionally contain at least one carbonyl group, L is oxygen or sulphur, R9 and R10 are each independently in each case optionally substituted alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, cycloalkyl, cycloalkyloxy, cycloalkenyloxy, cycloalkylalkoxy, alkylthio, alkenylthio, phenoxy, phenylthio, benzyloxy, benzylthio, heteroaryloxy, heteroarylthio, heteroarylalkoxy or heteroarylalkylthio, or R9 and R10 optionally form, together with the phosphorus atom to which they are bonded, a saturated or unsaturated and optionally substituted 5- to 7-membered ring which optionally contain one or two heteroatoms selected from the group consisting of oxygen (where oxygen atoms must not be immediately adjacent) and sulphur, and R11 and R12 are each independently in each case optionally substituted alkyl, alkenyl, alkynyl, phenyl or phenylalkyl, with the proviso that R7 in the group (F) is not methyl when G1 is C—H, G2 is the radical (A), R1 is methyl, n is 2, X is oxygen and A1, R2 and R6 are each hydrogen.
地址 Monheim am Rhein DE