发明名称 METHOD FOR THE PREPARATION OF 1-(2-HALOGEN-ETHYL)-4 PIPERIDINE-CARBOXYLIC ACID ETHYL ESTERS
摘要 The present invention refers to a process for the preparation of 1-(2-halogen-ethyl)-4-piperidinecarboxylic acid ethyl esters, in particular of 1-(2-chloroethyl)-4 piperidinecarboxylic acid ethyl ester, a versatile synthesis intermediate, particularly useful as an intermediate compound in the synthesis of umeclidinium.
申请公布号 WO2016071792(A1) 申请公布日期 2016.05.12
申请号 WO2015IB58145 申请日期 2015.10.22
申请人 LABORATORIO CHIMICO INTERNAZIONALE S.P.A. 发明人 BERTOLINI, GIORGIO;COLLI, CORRADO;BIANCHI, ALDO;COLOMBO, FEDERICA;MAIORANA, STEFANO;NISIC, FILIPPO
分类号 C07D211/52 主分类号 C07D211/52
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