发明名称 A PROCESS FOR PREPARATION OF (2S, 5R)-7-OXO-6-SULPHOOXY-2-[((3R)-PYRROLIDINE-3-CARBONYL)-HYDRAZINO CARBONYL]-1,6-DIAZA-BICYCLO[3.2.1]OCTANE
摘要 A process for preparation of (2S,5R)-7-oxo-6-sulphooxy-2-[((3R)-pyrrolidine-3-carbonyl)-hydrazino carbonyl]-1,6-diaza-bicyclo[3.2.1]octane is disclosed comprising reacting a compound of Formula (II) with a compound of Formula (III) to obtain a compound of Formula (IV). The crystalline end-product is als claimed.
申请公布号 EP3013830(A1) 申请公布日期 2016.05.04
申请号 EP20130812119 申请日期 2013.10.12
申请人 WOCKHARDT LIMITED 发明人 PAWAR, SHIVAJI SAMPATRAO;JADHAV, SUNIL BHAGINATH;MISHRA, AMIT CHANDRA;RANE, VIPUL;BHAWSAR, SATISH;DESHPANDE, PRASAD KESHAV;YEOLE, RAVINDRA DATTATRAYA;PATEL, MAHESH VITHALBHAI
分类号 C07D471/08 主分类号 C07D471/08
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