发明名称 BICYCLIC HETEROCYCLIC COMPOUNDS AS FGFR INHIBITORS
摘要 The invention relates to bicyclic heterocyclic derivative compounds, to pharmaceutical compositions comprising said compounds and to the use of said compounds in the treatment of cancer, proliferative disorders, or a disease state or condition mediated by a FGFR kinase, the compound having the structure of Formula (I). (see formula I)
申请公布号 CA2672172(C) 申请公布日期 2016.05.03
申请号 CA20072672172 申请日期 2007.12.21
申请人 ASTEX THERAPEUTICS LIMITED 发明人 BERDINI, VALERIO;BESONG, GILBERT EBAI;CALLAGHAN, OWEN;CARR, MARIA GRAZIA;CONGREVE, MILES STUART;GILL, ADRIAN LIAM;GRIFFITHS-JONES, CHARLOTTE MARY;MADIN, ANDREW;MURRAY, CHRISTOPHER WILLIAM;NIJJAR, RAJDEEP KAUR;O'BRIEN, MICHAEL ALISTAIR;PIKE, ANDREW;SAXTY, GORDON;TAYLOR, RICHARD DAVID;VICKERSTAFFE, EMMA
分类号 C07D471/04;A61K31/437;A61K31/519;A61P35/00;C07D487/04 主分类号 C07D471/04
代理机构 代理人
主权项
地址