发明名称 CRYSTALLINE FORM OF N,N-DICYCLOPROPYL-4-(1,5-DIMETHYL-1H-PYRAZOL-3-YLAMINO)-6-ETHYL-1-METHYL-1,6-DIHYDROIMIDAZO[4,5-D]PYRROLO[2,3-B]PYRIDINE-7-CARBOXAMIDE FOR THE TREATMENT OF MYELOPROLIFERATIVE DISORDERS
摘要 Crystalline form, Form HI.5-4, of N,N-di-cyclopropyl-4-(1,5-dimethyl-1H-pyrazol-3-ylamino)-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide, (Compound I) is provided. Also provided are a pharmaceutical composition and an oral dosage form comprising Form HI.5-4 of Compound I as well as a method of using the Form HI.5-4 of Compound I in the treatment of myeloproliferative disorders, which include polycythaemia vera, thrombocythaemia and primary myelofibrosis.
申请公布号 US2016115165(A1) 申请公布日期 2016.04.28
申请号 US201414892630 申请日期 2014.05.28
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 Tameze Shella
分类号 C07D471/16 主分类号 C07D471/16
代理机构 代理人
主权项 1. A crystalline form of Compound I:comprising Form H1.5-4.
地址 Princeton NJ US