Heterocyclic group contained amino-methanol derivative, and salt, synthetic method and use thereof

摘要

The present invention provides a heterocyclic group contained amino-methanol derivative, and salt, a preparation method and use thereof, and belongs to the medical field. The heterocyclic group contained amino-methanol derivative and the salt thereof of the present invention are used for preparing medicines for immune suppression and for the treatment of organ transplant rejection, or medicines for treating immune mediated inflammatory diseases, such as multiple sclerosis, systemic lupus erythematosus and rheumatoid arthritis.

主权项

1. A heterocyclic amino-methanol compound represented by the formula: wherein R1 is  where R5 is selected from the group consisting of alkyl, alkoxy and R7OCH2CH2O; R6 is selected from the group consisting of H, alkyl, ethoxy and fluoroalkyl; and R7 is alkyl; or a salt thereof.