发明名称 Análogos de buprenorfina como agonistas y/o antagonistas del receptor opioide
摘要 The present invention is directed to Buprenorphine Analog compounds of the Formula (I), Formula (IA) or Formula (IB) shown below, wherein R1, R2, R8, R3a, R 3b, G, X, Z and Y are as defined herein. Compounds of the Invention are useful for treating pain, constipation, and other conditions modulated by activity of opioid and ORL-1 receptors.
申请公布号 ES2566828(T3) 申请公布日期 2016.04.15
申请号 ES20110776855T 申请日期 2011.09.20
申请人 Purdue Pharma L.P. 发明人 KYLE, Donald J.;TAFESSE, Laykea
分类号 C07D489/12;A61K31/485;A61P25/04 主分类号 C07D489/12
代理机构 代理人
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