发明名称 |
TARTRATE SALT OF 5-CHLORO-THIOPHENE-2-CARBOXYLIC ACID [(S)-2-[METHYL-3-(2-OXO-PYRROLIDIN-1-YL)-BENZENESULFONYLAMINO]-3-(4-METHYL-PIPERAZIN-1-YL)-3-OXO-PROPYL]AMIDE |
摘要 |
The invention relates to the tartrate salt of 5-chloro-thiophene-2-carboxylic acid [(S)-2-[methyl-3-(2-oxo-pyrrolidin-1-yl) -benzenesulfonylamino]-3-(4-methyl-piperazin-1-yl)-3-oxo-propyl]amide, to its crystalline form, to its preparation and to its therapeutic use. |
申请公布号 |
US2016102082(A1) |
申请公布日期 |
2016.04.14 |
申请号 |
US201414786953 |
申请日期 |
2014.04.25 |
申请人 |
SANOFI |
发明人 |
Lafferrere Laurent;Villion Sebastien;Gauthier Sandrine;Bourbon Andre |
分类号 |
C07D409/14;C07C59/255 |
主分类号 |
C07D409/14 |
代理机构 |
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代理人 |
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主权项 |
1. An L-tartrate salt of 5-chloro-thiophene-2-carboxylic acid [(S)-2-[methyl-3-(2-oxo-pyrrolidin-1-yl)-benzenesulfonylamino]-3-(4-methyl-piperazin-1-yl)-3-oxo-propyl]amide. |
地址 |
Paris FR |