发明名称 TARTRATE SALT OF 5-CHLORO-THIOPHENE-2-CARBOXYLIC ACID [(S)-2-[METHYL-3-(2-OXO-PYRROLIDIN-1-YL)-BENZENESULFONYLAMINO]-3-(4-METHYL-PIPERAZIN-1-YL)-3-OXO-PROPYL]AMIDE
摘要 The invention relates to the tartrate salt of 5-chloro-thiophene-2-carboxylic acid [(S)-2-[methyl-3-(2-oxo-pyrrolidin-1-yl) -benzenesulfonylamino]-3-(4-methyl-piperazin-1-yl)-3-oxo-propyl]amide, to its crystalline form, to its preparation and to its therapeutic use.
申请公布号 US2016102082(A1) 申请公布日期 2016.04.14
申请号 US201414786953 申请日期 2014.04.25
申请人 SANOFI 发明人 Lafferrere Laurent;Villion Sebastien;Gauthier Sandrine;Bourbon Andre
分类号 C07D409/14;C07C59/255 主分类号 C07D409/14
代理机构 代理人
主权项 1. An L-tartrate salt of 5-chloro-thiophene-2-carboxylic acid [(S)-2-[methyl-3-(2-oxo-pyrrolidin-1-yl)-benzenesulfonylamino]-3-(4-methyl-piperazin-1-yl)-3-oxo-propyl]amide.
地址 Paris FR