发明名称 DERIVES DE GLYCOSIDES, LEUR PREPARATION ET LEUR UTILISATION COMME GROUPES PROSTHETIQUES
摘要 The present invention relates to glycoside-derived compounds, to the processes for preparing same and to the use thereof as prosthetic groups for radiolabelling biomolecules. These compounds are co-azido-alkyl 6-deoxy-6-[18F]-fluoroglycosides of formula (I), in which: k is equal to 2 or 3; n is an integer between 1 and 5; R is independently H or a C1-C5 alkyl group, m being an integer between 0 and 2 if k=2 and m between 0 and 3 if k=3; and X is chosen from the group comprising O, S, CH2 and NR′, in which R′ is independently a C1-C5 alkyl group or an aryl group, including all the stereoisomers thereof.
申请公布号 FR2992647(B1) 申请公布日期 2016.04.01
申请号 FR20120056308 申请日期 2012.07.02
申请人 CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE - CNRS;UNIVERSITE DE LORRAINE 发明人 CHAPLEUR YVES;LAMANDE SANDRINE;COLLET CHARLOTTE;CHRETIEN FRANCOISE
分类号 C07H5/02;A61K51/04 主分类号 C07H5/02
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