发明名称 Synthesis and novel salt forms of (r)-5-((e)-2-(pyrrolidin-3-ylvinyl)pyrimidine
摘要 Disclosed is a amorphous form of (R)-5-((E)-2-pyrrolidin-3-ylvinyl)pyrimidine mono-citrate. Also disclosed is the use of (R)-5-((E)-2-pyrrolidin-3-ylvinyl)pyrimidine mono-citrate for treating constipation.
申请公布号 NZ703381(A) 申请公布日期 2016.03.31
申请号 NZ20090703381 申请日期 2009.11.30
申请人 TARGACEPT INC. 发明人 AKIREDDY SRINIVISA RAO;MILLER CRAIG HARRISON;BHATTI BALWINDER SINGH;MUNOZ JULIO A;DULL GARY MAURICE;OTTEN PIETER ALBERT;MITCHENER JR. JOSEPH PIKE;CUTHBERTSON TIMOTHY J
分类号 C07D403/06;A61K31/505;A61P25/00 主分类号 C07D403/06
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