发明名称 |
Synthesis and novel salt forms of (r)-5-((e)-2-(pyrrolidin-3-ylvinyl)pyrimidine |
摘要 |
Disclosed is a amorphous form of (R)-5-((E)-2-pyrrolidin-3-ylvinyl)pyrimidine mono-citrate. Also disclosed is the use of (R)-5-((E)-2-pyrrolidin-3-ylvinyl)pyrimidine mono-citrate for treating constipation. |
申请公布号 |
NZ703381(A) |
申请公布日期 |
2016.03.31 |
申请号 |
NZ20090703381 |
申请日期 |
2009.11.30 |
申请人 |
TARGACEPT INC. |
发明人 |
AKIREDDY SRINIVISA RAO;MILLER CRAIG HARRISON;BHATTI BALWINDER SINGH;MUNOZ JULIO A;DULL GARY MAURICE;OTTEN PIETER ALBERT;MITCHENER JR. JOSEPH PIKE;CUTHBERTSON TIMOTHY J |
分类号 |
C07D403/06;A61K31/505;A61P25/00 |
主分类号 |
C07D403/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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