发明名称 CRYSTALLINE FORMS OF N,N-DICYCLOPROPYL-4-(1,5-DIMETHYL-1H-PYRAZOL-3-YLAMINO)-6-ETHYL-1-METHYL-1,6-DIHYDROIMIDAZO[4,5-D]PYRROLO[2,3-B]PYRIDINE-7-CARBOXIMIDE FOR THE TREATMENT OF MYELOPROLIFERATIVE DISORDERS
摘要 Crystalline form, Form T1H1.5-4, of N,N-dicyclopropyl-4-(1,5-dimethyl-1H-pyrazol-3-ylamino)-6-ethyl-1-methyl -1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide (Compound (I)) is provided. Also provided is a pharmaceutical composition and an oral dosage form comprising Form T1H1.5-4 of Compound (I) as well as a method of using the Form T1H1.5-4 of Compound for the treatment of myeloproliferative disorders, which include polycythaemia vera, thrombocythaemia and primary myelofibrosis.;
申请公布号 US2016090385(A1) 申请公布日期 2016.03.31
申请号 US201414892622 申请日期 2014.05.28
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 Purandare Ashok Vinayak;Wan Honghe
分类号 C07D471/14 主分类号 C07D471/14
代理机构 代理人
主权项 1. A crystalline form of Compound I: comprising Form T1H1.5-4.
地址 Princeton NJ US