PROCESSES FOR THE SYNTHESIS OF 5-(4-METHYL-1H-IMIDAZOL-1-YL)-3-(TRIFLUOROMETHYL)-BENZENAMINE AND ITS INTERMEDIATES
摘要
The present invention provides an efficient, safe and cost effective way to prepare 5-(4-methyl-1H-imidazol-1-yl)-3-(trifluoromethyl)-benzenamine which is a key intermediate for the preparation of substituted pyrimidinylaminobenzamides of formula (II). (see formula II)
申请公布号
CA2833394(C)
申请公布日期
2016.03.29
申请号
CA20062833394
申请日期
2006.06.07
申请人
NOVARTIS AG
发明人
ABEL, STEPHAN;ACEMOGLU, MURAT;ERB, BERNHARD;KRELL, CHRISTOPH;SCLAFANI, JOSEPH;MEISENBACH, MARK;PRASHAD, MAHAVIR;SHIEH, WEN-CHUNG;XUE, SONG