发明名称 AZA-ADAMANTANE DERIVATIVE MONOHYDRATE
摘要 FIELD: medicine, pharmaceutics.SUBSTANCE: invention refers to pharmaceutical composition modulating activity of α7 and/or α4β2 nicotinic acetylcholine receptors, containing a crystalline monohydrate of (4s)-4-(5-phenyl-1,3,4-thiadiazol-2-yloxy)-1-azatricyclo[3.3.1.1]decane dihydrocitrate as an active ingredient.EFFECT: using pharmaceutical composition containing a crystalline monohydrate of (4s)-4-(5-phenyl-1,3,4-thiadiazol-2-yloxy)-1-azatricyclo[3,3,1,1]decane dihydrocitrate having high stability and poor moisture absorption.3 cl, 9 dwg, 6 ex
申请公布号 RU2579121(C2) 申请公布日期 2016.03.27
申请号 RU20130118560 申请日期 2011.09.21
申请人 EBBVI BAKHAMAZ LTD. 发明人 CHEN SHUAN;NAPIR DZHEJMS DZH.;CHZHAN DZHEFF DZH. Z.;BREKMEJER POL DZH.
分类号 C07D471/18;A61K31/439;A61P25/00;A61P25/28 主分类号 C07D471/18
代理机构 代理人
主权项
地址