发明名称 METHOD OF PRODUCING PYRIPYROPENE DERIVATIVES
摘要 FIELD: chemistry.SUBSTANCE: invention relates to the method of producing the compound C:, which includes one- to three-step selective acylation of the hydroxyl group in the first position and in the eleventh position of the compound of formula B1:, with an acylating agent in a solvent selected from N-methyl-2-pyrrolidinone and N,N-dimethylacetamide, in the presence of a base selected from 2,4,6-collidine and 2,6-lutidine, or in the absence of a base.EFFECT: method enables to selectively obtain the compound C with high output.13 cl, 1 dwg, 5 tbl, 25 ex
申请公布号 RU2578605(C2) 申请公布日期 2016.03.27
申请号 RU20120141555 申请日期 2010.11.10
申请人 MEJDZI SEJKA FARMA KO., LTD. 发明人 FUKUDA JOSIMASA;ANDO TAKASI;GOTO KIMIKHIKO;NAKANISI NOZOMU;VATANABE TAKASI;KURIKHARA KENITI;MINOVA NOBUTO;MITOMI MASAAKI
分类号 C07D493/04 主分类号 C07D493/04
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