发明名称 |
Amorphous form of an AKT inhibiting pyrimidinyl-cyclopentane compound, compositions and methods thereof |
摘要 |
Disclosed is (S)-2-(4-chlorophenyl)-1-(4-((5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl)-3-(isopropylamino)propan-1-one monohydrochloride, forms, formulations, pharmaceutical compositions, processes of manufacturing and methods of use thereof. |
申请公布号 |
US9290458(B2) |
申请公布日期 |
2016.03.22 |
申请号 |
US201314401092 |
申请日期 |
2013.05.17 |
申请人 |
GENENTECH, INC. |
发明人 |
Chakravarty Paroma;Kothari Sanjeev;Gosselin Francis;Savage Scott J.;Stults Jeffrey |
分类号 |
C07D239/70;A61K31/496;C07D403/04;A61K31/517 |
主分类号 |
C07D239/70 |
代理机构 |
Viksnins Harris & Padys PLLP |
代理人 |
Viksnins Harris & Padys PLLP |
主权项 |
1. Amorphous (S)-2-(4-chlorophenyl)-1-(4-((5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl)-3-(isopropylamino)propan-1-one monohydrochloride. |
地址 |
South San Francisco CA US |