发明名称 Amorphous form of an AKT inhibiting pyrimidinyl-cyclopentane compound, compositions and methods thereof
摘要 Disclosed is (S)-2-(4-chlorophenyl)-1-(4-((5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl)-3-(isopropylamino)propan-1-one monohydrochloride, forms, formulations, pharmaceutical compositions, processes of manufacturing and methods of use thereof.
申请公布号 US9290458(B2) 申请公布日期 2016.03.22
申请号 US201314401092 申请日期 2013.05.17
申请人 GENENTECH, INC. 发明人 Chakravarty Paroma;Kothari Sanjeev;Gosselin Francis;Savage Scott J.;Stults Jeffrey
分类号 C07D239/70;A61K31/496;C07D403/04;A61K31/517 主分类号 C07D239/70
代理机构 Viksnins Harris & Padys PLLP 代理人 Viksnins Harris & Padys PLLP
主权项 1. Amorphous (S)-2-(4-chlorophenyl)-1-(4-((5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl)-3-(isopropylamino)propan-1-one monohydrochloride.
地址 South San Francisco CA US