发明名称 4-IMIDAZOPYRIDAZIN-1-YL-BENZAMIDES AND 4-IMIDAZOTRIAZIN-1-YL-BENZAMIDES AS BTK INHIBITORS
摘要 PROBLEM TO BE SOLVED: To provide compounds useful for the treatment of Brutons Tyrosine Kinase (Btk) mediated disorders.SOLUTION: The present invention relates to 6-5 membered fused pyridine ring compounds represented by the following formula.SELECTED DRAWING: None
申请公布号 JP2016034968(A) 申请公布日期 2016.03.17
申请号 JP20150202737 申请日期 2015.10.14
申请人 MERCK SHARP & DOHME BV 发明人 TJEERD A BARF;CHRISTIAAN GERARDUS JOHANNES MARIA JANS;DE ADRIANUS PETRUS ANTONIUS MAN;ARTHUR A OUBRIE;HANS C A RAAIJMAKERS;JOHANNES BERNARDUS MARIA REWINKEL;JAN-GERARD STERRENBURG;JACOBUS C H M WIJKMANS
分类号 C07D487/04;A61K31/4985;A61K31/506;A61K45/00;A61P43/00 主分类号 C07D487/04
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