发明名称 THIENOPYRIMIDINE INHIBITORS OF ATYPICAL PROTEIN KINASE C
摘要 The present application provides a compound of formula (I) or a salt thereof, wherein R1, R2, R3, R4, R5, R6, A, G, M, Q and X are as defined herein. A compound of formula (I) and its salts have aPKC inhibitory activity, and may be used to treat proliferative disorders.
申请公布号 EP2782917(B1) 申请公布日期 2016.03.02
申请号 EP20120795969 申请日期 2012.11.19
申请人 CANCER RESEARCH TECHNOLOGY LIMITED;IGNYTA, INC. 发明人 DORSEY, BRUCE D.;LEARN, KEITH S.;MORRIS, EMMA L.;OTT, GREGORY R.;ROFFEY, JONATHAN R.;SOUDY, CHRISTELLE N.;WAGNER, JASON C.
分类号 C07D495/04;A61K31/519;A61P35/00;C07D495/14 主分类号 C07D495/04
代理机构 代理人
主权项
地址