发明名称 |
THIENOPYRIMIDINE INHIBITORS OF ATYPICAL PROTEIN KINASE C |
摘要 |
The present application provides a compound of formula (I) or a salt thereof, wherein R1, R2, R3, R4, R5, R6, A, G, M, Q and X are as defined herein. A compound of formula (I) and its salts have aPKC inhibitory activity, and may be used to treat proliferative disorders. |
申请公布号 |
EP2782917(B1) |
申请公布日期 |
2016.03.02 |
申请号 |
EP20120795969 |
申请日期 |
2012.11.19 |
申请人 |
CANCER RESEARCH TECHNOLOGY LIMITED;IGNYTA, INC. |
发明人 |
DORSEY, BRUCE D.;LEARN, KEITH S.;MORRIS, EMMA L.;OTT, GREGORY R.;ROFFEY, JONATHAN R.;SOUDY, CHRISTELLE N.;WAGNER, JASON C. |
分类号 |
C07D495/04;A61K31/519;A61P35/00;C07D495/14 |
主分类号 |
C07D495/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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