摘要 |
THE INVENTION RELATES TO SUBSTITUTED NITROGEN CONTAINING BICYCLIC HETEROCYCLES OF THE FORMULA (I): WHEREIN Z IS CH? OR N-R? AND X, R¹, R², R?, R?, R? AND N ARE AS DEFINED IN THE DESCRIPTION. SUCH COMPOUNDS ARE SUITABLE FOR THE TREATMENT OF A DISORDER OR DISEASE WHICH IS MEDIATED BY THE ACTIVITY OF MDM2 AND/OR MDM4, OR VARIANTS THEREOF. |
申请人 |
NOVARTIS AG |
发明人 |
BERGHAUSEN,JOERG;PISSOT SOLDERMANN,CAROLE;REN,HAIXIA;STUTZ,STEFAN;BUSCHMANN,NICOLE;FURET,PASCAL;GESSIER,FRANÇOIS;HERGOVICH LISZTWAN,JOANNA;HOLZER,PHILIPP;JACOBY,EDGAR;KALLEN,JOERG;MASUYA,KEIICHI |