发明名称 ACTIVE METABOLITE OF 1-[(2-BROMOPHENYL) SULFONYL]-5-METHOXY-3- [(4-METHYL-1-PIPERAZINYL) METHYL]-1H-INDOLE DIMESYLATE MONOHYDRATE AND DIMESYLATE DIHYDRATE SALT OF ACTIVE METABOLITE
摘要 The present invention is directed to active metabolite of 1-[(2- bromophenyl)sulfonyl]-5-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole dimesylate monohydrate having the following structure The present invention is also directed to dimesylate dihydrate salt of formula (I) having the following structure The compounds of formula (I) and formula (II) are useful in the treatment of various disorders that are related to 5-HT6 receptor antagonist.
申请公布号 CA2957497(A1) 申请公布日期 2016.02.25
申请号 CA20142957497 申请日期 2014.10.20
申请人 SUVEN LIFE SCIENCES LIMITED 发明人 NIROGI, RAMAKRISHNA;KAMBHAMPATI, RAMASASTRI;SHINDE, ANIL KARBHARI;JASTI, VENKATESWARLU
分类号 A61K31/4045;A61P25/00;C07D209/14 主分类号 A61K31/4045
代理机构 代理人
主权项
地址