发明名称 POLYCYCLIC PYRIDONE DERIVATIVE HAVING INTEGRASE-INHIBITING ACTIVITY
摘要 The present invention relates to: a novel compound having an anti-viral activity, more specifically a pyridone derivative having an HIV integrase-inhibiting activity; and a medicine, specifically an anti-HIV drug, which contains the compound or the pyridone derivative. The compound according to the present invention has an activity of inhibiting integrase in a virus, particularly an HIV and a resistant HIV and/or an activity of inhibiting the proliferation of cells of the virus. Therefore, the compound is useful for the prevention or treatment of various integrase-related diseases, viral infections (e.g., AIDS) and others.
申请公布号 WO2016027879(A1) 申请公布日期 2016.02.25
申请号 WO2015JP73487 申请日期 2015.08.21
申请人 SHIONOGI & CO., LTD. 发明人 YOSHINAGA, TOMOKAZU;NODU, KOUHEI
分类号 C07D471/04;A61K31/4985;A61K31/519;A61K31/53;A61K31/5365;A61K31/553;A61P31/18;A61P43/00;C07D471/14;C07D471/22;C07D498/14 主分类号 C07D471/04
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