发明名称 PROCESSES FOR THE PREPARATION OF A BACE INHIBITOR
摘要 This invention provides processes for the preparation of verubecestat (Compound of Formula (I)), a potent inhibitor of BACE-1 and BACE-2. In addition, the invention provides certain synthetic intermediates which are useful, among other things, for the preparation of the Compound of Formula (I).
申请公布号 WO2016025359(A1) 申请公布日期 2016.02.18
申请号 WO2015US44410 申请日期 2015.08.10
申请人 MERCK SHARP & DOHME CORP.;MILLER, STEVEN, P.;MOLINARO, CARMELA;THAISRIVONGS, DAVID;XU, FENG;DESMOND, RICHARD;LI, HONGMING;CHEN, QINGHAO;STAMFORD, ANDREW;SONG, ZHIGUO JAKE;TAN, LUSHI 发明人 MILLER, STEVEN, P.;MOLINARO, CARMELA;THAISRIVONGS, DAVID;XU, FENG;DESMOND, RICHARD;LI, HONGMING;CHEN, QINGHAO;STAMFORD, ANDREW;SONG, ZHIGUO JAKE;TAN, LUSHI
分类号 A61K31/549;C07D213/75;C07D417/02 主分类号 A61K31/549
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