发明名称 |
PROTEIN KINASE C INHIBITORS AND METHODS OF THEIR USE |
摘要 |
PKC inhibitors are disclosed. The PKC inhibitors are useful for treating PKC associated diseases, including certain cancers. The PKC inhibitors have improved efficacy at lower dosage amounts to achieve tumor regression, improved potency, PK profile, absorption, gastrointestinal tolerance and kinase selectivity. |
申请公布号 |
WO2016020864(A1) |
申请公布日期 |
2016.02.11 |
申请号 |
WO2015IB55951 |
申请日期 |
2015.08.05 |
申请人 |
NOVARTIS AG;LUZZIO, MICHAEL JOSEPH;PAPILLON, JULIEN;VISSER, MICHAEL SCOTT |
发明人 |
LUZZIO, MICHAEL JOSEPH;PAPILLON, JULIEN;VISSER, MICHAEL SCOTT |
分类号 |
C07D401/14;A61K31/506;A61P31/04;C07D413/14 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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