发明名称 CRYSTALLINE FORMS OF CANAGLIFLOZIN
摘要 The present invention relates to crystalline forms of canagliflozin, processes for their preparation, and their use for the treatment of type 2 diabetes mellitus. A crystalline Form R1of canagliflozin emihydrate. The crystalline Form R1 of canagliflozin hemihydrate of claim 1, characterized by an X-ray powder diffraction peaks having d-spacing values at about 3.1, 3.7, 4.6, and 8.9 A.
申请公布号 WO2016016774(A1) 申请公布日期 2016.02.04
申请号 WO2015IB55559 申请日期 2015.07.22
申请人 SUN PHARMACEUTICAL INDUSTRIES LIMITED 发明人 SANTRA, RAMKINKAR;NAGDA, DEVENDRA, PRAKASH;THAIMATTAM, RAM;ARYAN, SATISH, KUMAR;SINGH, TARUN, KUMAR;PRASAD, MOHAN;GANGULY, SOMENATH;WADHWA, DEEPIKA
分类号 C07D409/10 主分类号 C07D409/10
代理机构 代理人
主权项
地址