发明名称 GLYCOSIDE DERIVATIVES, PREPARATION THEREOF AND USE THEREOF AS PROSTHETIC GROUPS
摘要 The present invention relates to glycoside-derived compounds, to the processes for preparing same and to the use thereof as prosthetic groups for radiolabelling biomolecules. These compounds are co-azido-alkyl 6-deoxy-6-[18F]-fluoroglycosides of formula (I), in which: k is equal to 2 or 3; n is an integer between 1 and 5; R is independently H or a C1-C5 alkyl group, m being an integer between 0 and 2 if k=2 and m between 0 and 3 if k=3; and X is chosen from the group comprising O, S, CH2 and NR′, in which R′ is independently a C1-C5 alkyl group or an aryl group, including all the stereoisomers thereof.;
申请公布号 US2016031923(A1) 申请公布日期 2016.02.04
申请号 US201314412161 申请日期 2013.07.02
申请人 UNIVERSITÉ DE LORRAINE ;CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE - CNRS 发明人 CHAPLEUR YVES;LAMANDE Sandrine;COLLET Charlotte;CHRETIEN Françoise
分类号 C07H15/04 主分类号 C07H15/04
代理机构 代理人
主权项
地址 Nancy Cedex FR