发明名称 BENZIMIDAZOLONE DERIVATIVES AS BROMODOMAIN INHIBITORS
摘要 This application relates to chemical compounds which may act as inhibitors of, or which may otherwise modulate the activity of, a bromodomain-containing protein, including bromodomain-containing protein 4 (BRD4), and to compositions and formulations containing such compounds, and methods of using and making such compounds. Compounds include compounds of Formula (I) wherein R1a, R1b, R2a, R2b, R3, and X are described herein.
申请公布号 EP2978759(A1) 申请公布日期 2016.02.03
申请号 EP20140729114 申请日期 2014.03.27
申请人 GILEAD SCIENCES, INC. 发明人 AKTOUDIANAKIS, EVANGELOS;CHIN, GREGORY;CORKEY, BRITTON KENNETH;DU, JINFA;ELBEL, KRISTYNA;JIANG, ROBERT H.;KOBAYASHI, TETSUYA;MARTINEZ, RUBEN;METOBO, SAMUEL E.;MISH, MICHAEL;SHEVICK, SOPHIE;SPERANDIO, DAVID;YANG, HAI;ZABLOCKI, JEFF
分类号 C07D413/14;A61K31/42;A61P35/00;C07D413/04;C07D417/14 主分类号 C07D413/14
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