发明名称 |
PROCESS FOR THE MANUFACTURE OF (R)-5-[2-(5,6-DIETHYLINDAN-2-YLAMINO)-1-HYDROXYETHYL]-8-HYDROXY-(1H)-QUINOLIN-2-ONE |
摘要 |
The present invention provides an efficient process for manufacturing (R)-5-[2-(5,6-diethyl-indan-2-yl-amino)-1-hydroxyethyl]-8-hydroxy-(1H)-quinolin-2-one, commonly known as indacaterol, or a pharmaceutically acceptable salt thereof, comprising intermediates of synthesis of Formula (II) and Formula (III). |
申请公布号 |
EP2978745(A1) |
申请公布日期 |
2016.02.03 |
申请号 |
EP20140712694 |
申请日期 |
2014.03.27 |
申请人 |
LABORATORIOS LESVI, S.L. |
发明人 |
DALMASES BARJOAN, PERE;HUGUET CLOTET, JUAN;CAPDEVILA URBANEJA, ENRIC |
分类号 |
C07D215/26 |
主分类号 |
C07D215/26 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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