发明名称 A PROCESS FOR PREPARATION OF ANAGLIPTIN HYDROCHLORIDE
摘要 <p>The present invention relates to process for preparing dipeptidyl peptidase IV inhibitor Anagliptin free base or its hydrochloride salt by using novel methane sulfonic acid salt of (2S)-1-{[(1-Amino-2-methylpropan-2-yl) amino] acetyl} pyrrolidine-2-carbonitrile (formula IIa). Anagliptin is used for the treatment of diabetes.</p>
申请公布号 WO2016012927(A1) 申请公布日期 2016.01.28
申请号 WO2015IB55481 申请日期 2015.07.20
申请人 LUPIN LIMITED 发明人 ANSARI, SHAHID, AKHTAR;YADAV, ASHOK, KESHAVLAL;PATIL, TUSHAR, YASHWANT;PATHAK, DHARMENDRAKUMAR, SHRIPATI;BARIA, REENABEN, RATANSING;PATIL, SHASHIKANT, PRABHAKAR
分类号 C07D487/04;A61K31/519;A61P3/10;C07D207/09 主分类号 C07D487/04
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