发明名称 |
SMALL MOLECULE TRANSCRIPTION MODULATORS OF BROMODOMAINS |
摘要 |
This disclosure relates generally to compounds and compositions comprising one or more indole analogs. These compounds are useful for treating diseases associated with NF-kB and p53 activity, such as cancer and inflammatory diseases. |
申请公布号 |
WO2015184257(A3) |
申请公布日期 |
2016.01.21 |
申请号 |
WO2015US33178 |
申请日期 |
2015.05.29 |
申请人 |
ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI |
发明人 |
ZHOU, MING-MING;GERONA-NAVARRO, GUILLERMO;RODRIGUEZ-FERNANDEZ, YOEL;CASACCIA, PATRIZIA |
分类号 |
A61K31/497;A01N43/38;A01N43/42;C07D217/00;C07D487/00 |
主分类号 |
A61K31/497 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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