发明名称 PRODRUG DERIVATIVES OF (E)-N-METHYL-N-((3-METHYLBENZOFURAN-2-YL)METHYL)-3-(7-OXO-5,6,7,8-TETRAHYDRO-1,8-NAPHTHYRIDIN-3-YL)ACRYLAMIDE
摘要 In part, the present disclosure is directed to prodrug derivatives of (E)-N-methyl-N-((3-methylbenzofuran-2-yl)methyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamide compounds with significant solubility and bioavailability profiles.
申请公布号 EP2861608(A4) 申请公布日期 2016.01.20
申请号 EP20130806968 申请日期 2013.06.19
申请人 DEBIOPHARM INTERNATIONAL SA 发明人 PARTRIDGE, JOHN, J.;COLUCCI, JOHN;GAREAU, YVES;THERIEN, MICHEL;ZAMBONI, ROBERT;HAFKIN, BARRY;MARFAT, ANTHONY;ZAGHDANE, HELMI
分类号 C07F9/6561;A61K31/675;A61P31/04;C07F9/60 主分类号 C07F9/6561
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