发明名称 |
TRIAZOLOPYRIDINES AND TRIAZOLOPYRAZINES AS LSD1 INHIBITORS |
摘要 |
<p>The present invention is directed to [1,2,4]triazolo[4,3-a]pyridine and [1,2,4]triazolo[4,3-a]pyrazine derivatives which are LSD1 inhibitors useful in the treatment of diseases such as cancer.</p> |
申请公布号 |
WO2016007727(A1) |
申请公布日期 |
2016.01.14 |
申请号 |
WO2015US39718 |
申请日期 |
2015.07.09 |
申请人 |
INCYTE CORPORATION |
发明人 |
WU, LIANGXING;SUN, YAPING;WANG, XIAOZHAO;YAO, WENQING;ZHANG, COLIN |
分类号 |
C07D471/04;A61K31/437;A61K31/4985;A61P35/00;C07D487/04 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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