发明名称 |
CHEMICAL COMPOUND USEFUL AS INTERMEDIATE FOR PREPARING A CATECHOL-O-METHYLTRANSFERASE INHIBITOR |
摘要 |
There is disclosed a methylated intermediate which may be demethylated to provide an inhibitor of catechol-O-methyltransferase useful in the treatment of Parkinson's disease. Also disclosed are methods of making and using said intermediate. |
申请公布号 |
US2016009700(A1) |
申请公布日期 |
2016.01.14 |
申请号 |
US201514814603 |
申请日期 |
2015.07.31 |
申请人 |
BIAL - Portela & Cª., S.A |
发明人 |
Russo Domenico;Kiss Laszlo Erno;Wahnon Jorge Bruno Reis;Learmonth David Alexander;Eszenyi Tibor;Zimmermann Axel;Schlummer Bjoern;Kreis Michael;Reiter Klaus |
分类号 |
C07D413/04 |
主分类号 |
C07D413/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
S. Mamede Do Coronado PT |