发明名称 |
AMORPHOUS FORM OF 4-((4-(CYCLOPENTYLOXY)-5-(2-METHYLBENZO[D]OXAZOL-6-YL)-7H-PYRROLO[2,3-D]PYRIMIDIN-2-YL)AMINO)-3-METHOXY-N-METHYLBENZAMIDE, COMPOSITIONS THEREOF AND METHODS OF THEIR USE |
摘要 |
Provided herein is an amorphous form of 4-((4-(Cyclopentyloxy)-5-(2-methylbenzo[d]oxazol-6-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)-3-methoxy-N-methylbenzamide, compositions thereof, and methods of their use for treating or preventing a cancer, in particular solid tumors and hematological cancers as described herein. |
申请公布号 |
US2016009722(A1) |
申请公布日期 |
2016.01.14 |
申请号 |
US201514797542 |
申请日期 |
2015.07.13 |
申请人 |
Signal Pharmaceuticals, LLC |
发明人 |
CHEN Ming J.;MUSLEHIDDINOGLU Jale;RUCHELMAN Alexander;Connolly Terrence Joseph |
分类号 |
C07D487/04 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
1. An amorphous form comprising Compound 1, or a tautomer thereof: |
地址 |
San Diego CA US |