发明名称 AMORPHOUS FORM OF 4-((4-(CYCLOPENTYLOXY)-5-(2-METHYLBENZO[D]OXAZOL-6-YL)-7H-PYRROLO[2,3-D]PYRIMIDIN-2-YL)AMINO)-3-METHOXY-N-METHYLBENZAMIDE, COMPOSITIONS THEREOF AND METHODS OF THEIR USE
摘要 Provided herein is an amorphous form of 4-((4-(Cyclopentyloxy)-5-(2-methylbenzo[d]oxazol-6-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl)amino)-3-methoxy-N-methylbenzamide, compositions thereof, and methods of their use for treating or preventing a cancer, in particular solid tumors and hematological cancers as described herein.
申请公布号 US2016009722(A1) 申请公布日期 2016.01.14
申请号 US201514797542 申请日期 2015.07.13
申请人 Signal Pharmaceuticals, LLC 发明人 CHEN Ming J.;MUSLEHIDDINOGLU Jale;RUCHELMAN Alexander;Connolly Terrence Joseph
分类号 C07D487/04 主分类号 C07D487/04
代理机构 代理人
主权项 1. An amorphous form comprising Compound 1, or a tautomer thereof:
地址 San Diego CA US