发明名称 |
Manufacture of 2-(5-bromo-4(-cyclopropylnaphthalen-1-yl)-4h-1,2,4-triazol-3-ylthio)acetic acid |
摘要 |
<p>Disclosed is processes for the synthesis of 2-(S-bromo-4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-yl-thio)acetic acid (compound of formula III) comprising brominating a precursor compound with N-bromosuccinimide (NBS) and a solvent.</p> |
申请公布号 |
NZ631044(A) |
申请公布日期 |
2015.12.24 |
申请号 |
NZ20130631044 |
申请日期 |
2013.07.02 |
申请人 |
ARDEA BIOSCIENCES INC. |
发明人 |
GUNIC ESMIR;GALVIN GABRIEL |
分类号 |
C07D249/12;A61K31/4196;A61P9/00;A61P29/00 |
主分类号 |
C07D249/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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