发明名称 |
HETEROCYCLIC AMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS |
摘要 |
<p>The invention relates to heterocyclic amide derivatives of formula (I), wherein R1, R2, R3, X and n are as defined in the description, their preparation and their use as pharmaceutically active compounds.</p> |
申请公布号 |
EP2804865(B1) |
申请公布日期 |
2015.12.23 |
申请号 |
EP20130707053 |
申请日期 |
2013.01.18 |
申请人 |
ACTELION PHARMACEUTICALS LTD. |
发明人 |
HILPERT, KURT;HUBLER, FRANCIS;KIMMERLIN, THIERRY;RENNEBERG, DORTE;STAMM, SIMON |
分类号 |
C07D491/048;A61K31/4355;A61P29/00 |
主分类号 |
C07D491/048 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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