发明名称 |
ALBICIDIN DERIVATIVES, THEIR USE AND SYNTHESIS |
摘要 |
Antibiotically active compounds characterized by general formula (I), wherein X1, BB, BC, BD, BE and X2 are building blocks with D1, D2, D3, D4 or D5 being linkers which include carbon, sulphur, nitrogen, phosphor and/or oxygen atoms and which are covalently connecting the moities BA and BB, BB and BC, BC and BD, BD and BE and BE and BF, respectively, and wherein in particular the building block BC comprises an amino acid derivative. The compounds for use in a method of treatment of diseases, in particular for use in a method of treatment of bacterial infections are also disclosed. |
申请公布号 |
EP2956437(A1) |
申请公布日期 |
2015.12.23 |
申请号 |
EP20140712606 |
申请日期 |
2014.02.14 |
申请人 |
CENTRE DE COOPERATION INTERNATIONALE EN RECHERCHEAGRONOMIQUE POUR LE DEVELOPPEMENT |
发明人 |
SÜSSMUTH, RODERICH;KRETZ, JULIAN;SCHUBERT, VIVIEN;PESIC, ALEXANDER;HÜGELLAND, MANUELA;ROYER, MONIQUE;COCIANCICH, STÉPHANE;ROTT, PHILIPPE;KERWAT, DENNIS;GRÄTZ, STEFAN |
分类号 |
C07C255/57;A61K31/277;A61K31/5375;A61P31/04;C07C233/83;C07C255/03;C07C311/21;C07D207/34;C07D241/28;C07D277/56;C07D295/14;C07D307/56;C07D317/08;C07D333/38;C07F9/09 |
主分类号 |
C07C255/57 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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