发明名称 |
FUSED BICYCLIC HETEROAROMATIC DERIVATIVES AS KINASE INHIBITORS |
摘要 |
<p>A series of fused bicyclic heteroaromatic derivatives of formula (IA) or (IB), as defined herein, being selective inhibitors of phosphatidylinositol-4-kinase IIIβ (PI4KIIIβ) activity, are beneficial in the treatment and/or prevention of various human ailments, including inflammatory, autoimmune and oncological disorders; viral diseases and malaria; and organ and cell transplant rejection.</p> |
申请公布号 |
WO2015193168(A1) |
申请公布日期 |
2015.12.23 |
申请号 |
WO2015EP63051 |
申请日期 |
2015.06.11 |
申请人 |
UCB BIOPHARMA SPRL;KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D |
发明人 |
FORD, DANIEL JAMES;HUANG, QIUYA;NEUSS, JUDI CHARLOTTE;REUBERSON, JAMES THOMAS;VANDERHOYDONCK, BART |
分类号 |
C07D487/04;A61K31/519;A61P29/00;A61P35/00;C07D495/04;C07D498/04 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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