发明名称 |
Formoterol, eventuelt farmak. kompat. Syreaddisjons-salter derav, spes. formoterolfumarat samt 3(R)-(22-hydroksy-2,2-ditien-2-ylacetoksy)-1-(3-fenoksypropyl)-1-azoniabicyklo[2.2,2]oktan som et salt med anion X som er et farm. aksept. anion av monovalent/polyvalent syre (INN aklidinium), spes. 3(R)-(2-hydroksy-2,2-ditien-2-ylacetoksy)-1-(3-fenoksypropyl)-1-azoniabicyklo[2.2.2]oktanbromid |
摘要 |
<p>Combination (I) comprises a phosphodiesterase inhibitor 4 (PDE4) (A) and an antagonist of M3 muscarinic receptors (B) (3(R)-(2-hydroxy-2, 2-dithien-2-ylacetoxy)-1-(3-phenoxypropyl)-1-azoniabicyclo [2.2.2] octane), in the form of a salt having an anion X (anion of a mono or polyvalent acid). An independent claim is also included for a method of treating a patient suffering from or susceptible to a respiratory disease or condition which responds to M3 antagonism comprising simultaneous, concurrent, separate or sequential administration of (I). ACTIVITY : Antiasthmatic; Respiratory-Gen.; Antiinflammatory. MECHANISM OF ACTION : Phosphodiesterase-4 inhibitor; Muscarinic receptors antagonist; Leukotriene-D4 antagonist; Neurokinin-1- receptor antagonist; Epidermal growth factor receptor kinase inhibitor; Beta-2 agonist; p38 Kinase inhibitor.</p> |
申请公布号 |
NO2015007(I2) |
申请公布日期 |
2015.12.21 |
申请号 |
NO20150000007C |
申请日期 |
2015.02.27 |
申请人 |
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发明人 |
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分类号 |
A61K31/137;A61K31/167;A61K31/439;A61K31/573;A61K31/58;A61K31/655;A61K45/00;A61K45/06 |
主分类号 |
A61K31/137 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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