发明名称 IMIDAZOPYRIDAZINE DERIVATIVES AS MODULATORS OF THE GABAA RECEPTOR ACTIVITY.
摘要 The present invention relates to imidazopyridazine derivatives. More particularly, it relates to 4-(biphenyl-3-yl)-7H-imidazo[4,5-c]pyridazine derivatives of formula (I) and pharmaceutically acceptable salts thereof, wherein R1, R2, R3, R4, R and R6 are as defined in the description. The imidazopyridazine derivatives of the present invention modulate the activity of the GABAA receptor. They are useful in the treatment of a number of conditions, including pain.
申请公布号 WO2015189744(A1) 申请公布日期 2015.12.17
申请号 WO2015IB54200 申请日期 2015.06.03
申请人 PFIZER LIMITED 发明人 OWEN, ROBERT MCKENZIE;PRYDE, DAVID CAMERON;TAKEUCHI, MIFUNE;WATSON, CHRISTINE ANNE LOUISE
分类号 C07D487/04;A61K31/5025;A61P25/00 主分类号 C07D487/04
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