发明名称 CHIRAL AMINES, A PROCESS FOR PREPARATION AND USE THEREOF
摘要 Described herein is the general synthesis of chiral amine from vinyl nitro compounds using Josiphos catalyst. The process is applied to develop a novel route to Sitagliptin (a DPP-IV inhibitor).
申请公布号 WO2015189862(A1) 申请公布日期 2015.12.17
申请号 WO2015IN50040 申请日期 2015.06.03
申请人 COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH 发明人 BARUA, NABIN CHANDRA;SAIKIA, BISHWAJIT;BORAH, PREETISMITA;BAISHYA, GAKUL
分类号 C07C227/18;C07B53/00;C07C201/12;C07C227/32;C07C229/08;C07C229/34;C07D487/04 主分类号 C07C227/18
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