发明名称 |
SUPER LEWIS ACIDIC BORATE ESTERS AS 18F-LABELED PET PROBES |
摘要 |
Compounds having a 1-bora-1-fluoro-2,6,7-trioxabicyclo[2.2.2]octane moiety wherein the fluorine is 18F are described. Also described are reagents for radiolabeling a molecule having Formula I. Method for radiolabeling molecules with the disclosed reagents are also descried, as are radiolabeled molecules prepared thereby. |
申请公布号 |
US2015361110(A1) |
申请公布日期 |
2015.12.17 |
申请号 |
US201414762544 |
申请日期 |
2014.01.24 |
申请人 |
UNIVERSITY OF SOUTH FLORIDA ;H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. |
发明人 |
McLaughlin Mark Lee;Tian Haibin |
分类号 |
C07F5/04;C07K7/56;C07B59/00 |
主分类号 |
C07F5/04 |
代理机构 |
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代理人 |
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主权项 |
1. A compound having the following moiety: wherein the fluorine is 18F. |
地址 |
Tampa FL US |