发明名称 N-AROYL CYCLIC AMINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS
摘要 Disclosed are N-aroyl cyclic amine derivatives having the formula: where the variables are as define herein, and their use as pharmaceuticals, specifically as orexin receptor antagonists.
申请公布号 US2009012122(A1) 申请公布日期 2009.01.08
申请号 US20070928072 申请日期 2007.10.30
申请人 SMITHKLINE BEECHAM P.L.C. 发明人 BRANCH CLIVE LESLIE;CHAN WAI NGOR;JOHNS AMANDA;JOHNSON CHRISTOPHER NORBERT;NASH DAVID JOHN;NOVELLI RICCARDO;PILLEUX JEAN-PIERRE;PORTER RODERICK ALAN;STEAD RACHEL ELIZABETH, ANNE;STEMP GEOFFREY
分类号 A61K31/454;C07D491/048;A61K31/4184;A61K31/426;A61K31/453;A61K31/4545;A61K31/4709;A61K31/496;A61K31/506;A61K31/5377;A61P1/04;A61P1/08;A61P1/14;A61P3/04;A61P3/10;A61P5/02;A61P5/10;A61P5/38;A61P7/00;A61P9/02;A61P9/04;A61P9/12;A61P11/06;A61P13/08;A61P13/10;A61P13/12;A61P15/00;A61P19/10;A61P25/00;A61P25/02;A61P25/04;A61P25/06;A61P25/08;A61P25/14;A61P25/16;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P35/00;A61P37/08;C07D401/06;C07D401/14;C07D403/14;C07D405/06;C07D405/14;C07D409/14;C07D413/14;C07D417/04;C07D417/14;C07D471/04;C07D491/04 主分类号 A61K31/454
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