发明名称 |
N-AROYL CYCLIC AMINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS |
摘要 |
Disclosed are N-aroyl cyclic amine derivatives having the formula: where the variables are as define herein, and their use as pharmaceuticals, specifically as orexin receptor antagonists.
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申请公布号 |
US2009012122(A1) |
申请公布日期 |
2009.01.08 |
申请号 |
US20070928072 |
申请日期 |
2007.10.30 |
申请人 |
SMITHKLINE BEECHAM P.L.C. |
发明人 |
BRANCH CLIVE LESLIE;CHAN WAI NGOR;JOHNS AMANDA;JOHNSON CHRISTOPHER NORBERT;NASH DAVID JOHN;NOVELLI RICCARDO;PILLEUX JEAN-PIERRE;PORTER RODERICK ALAN;STEAD RACHEL ELIZABETH, ANNE;STEMP GEOFFREY |
分类号 |
A61K31/454;C07D491/048;A61K31/4184;A61K31/426;A61K31/453;A61K31/4545;A61K31/4709;A61K31/496;A61K31/506;A61K31/5377;A61P1/04;A61P1/08;A61P1/14;A61P3/04;A61P3/10;A61P5/02;A61P5/10;A61P5/38;A61P7/00;A61P9/02;A61P9/04;A61P9/12;A61P11/06;A61P13/08;A61P13/10;A61P13/12;A61P15/00;A61P19/10;A61P25/00;A61P25/02;A61P25/04;A61P25/06;A61P25/08;A61P25/14;A61P25/16;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P35/00;A61P37/08;C07D401/06;C07D401/14;C07D403/14;C07D405/06;C07D405/14;C07D409/14;C07D413/14;C07D417/04;C07D417/14;C07D471/04;C07D491/04 |
主分类号 |
A61K31/454 |
代理机构 |
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代理人 |
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