发明名称 |
HETEROBICYCLIC COMPOUNDS AS GLUCOKINASE ACTIVATORS |
摘要 |
Compounds of Formula (I): wherein R1 to R11, A and X1 to X3 are as described in the specification, and their salts, are activators of glucokinase (GLK) and are thereby useful in the treatment of, for example, type 2 diabetes. Processes for preparing compounds of Formula (I) are also described.
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申请公布号 |
US2009105263(A1) |
申请公布日期 |
2009.04.23 |
申请号 |
US20060066967 |
申请日期 |
2006.09.12 |
申请人 |
CAULKETT PETER WILLIAM RODNEY;MCKERRECHER DARREN;NEWCOMBE NICHOLAS JOHN;PIKE KURT GORDON;ROBB GRAEME RICHARD;WARING MICHAEL JAMES |
发明人 |
CAULKETT PETER WILLIAM RODNEY;MCKERRECHER DARREN;NEWCOMBE NICHOLAS JOHN;PIKE KURT GORDON;ROBB GRAEME RICHARD;WARING MICHAEL JAMES |
分类号 |
A61K31/4985;A61K31/437;A61K31/519;C07D471/04;C07D487/04 |
主分类号 |
A61K31/4985 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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