发明名称 |
SOLID FORMS OF EMTRICITABINE |
摘要 |
The present invention provides novel crystalline forms of Emtricitabine, designated Emtricitabine form ULT-I, form ULT-2 and ULT-3, methods for the preparation of Emtricitabine form ULT-I, ULT-2 and ULT-3 and the use of Emtricitabine form ULT-I and/or ULT-2 and/or ULT-3 in pharmaceutical applications, in particular in anti-HIV medicaments. The crystalline form of Emtricitabine form ULT-I, ULT-2 and/or ULT-3 can be used in combination with other anti-HIV medicaments such as Efavirenz and Tenofovir DF. |
申请公布号 |
WO2009005338(A2) |
申请公布日期 |
2009.01.08 |
申请号 |
WO2008NL00158 |
申请日期 |
2008.06.23 |
申请人 |
ULTIMORPHIX TECHNOLOGIES B.V.;DOVA, EVANTHIA;VAN DER PLOEG, IDA |
发明人 |
DOVA, EVANTHIA;VAN DER PLOEG, IDA |
分类号 |
C07D411/04;A61K31/506;A61P31/18 |
主分类号 |
C07D411/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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