发明名称 Peptidase Inhibitors
摘要 The present invention relates to a series of novel compounds having the formula (I) wherein: X is NR<SUP>3 </SUP>or O; n is 1 or 2; A is a bicyclic carbocycle and R1 and R2 are as described herein. The compounds are useful as DPP-IV inhibitors, such as for the treatment of diabetes.
申请公布号 US2008234292(A1) 申请公布日期 2008.09.25
申请号 US20050571857 申请日期 2005.07.21
申请人 ROYALTY SUSAN MARIE;BURNS JAMES FORD;SCICINSKI JAN JOZEF;JAGDMANN JR GUNNAR ERIK;FOGLESONG ROBERT JAMES;RING KELLEE GRIFFIN;DYAKONOV TATYANA;MIDDLEMISS DAVID 发明人 ROYALTY SUSAN MARIE;BURNS JAMES FORD;SCICINSKI JAN JOZEF;JAGDMANN, JR. GUNNAR ERIK;FOGLESONG ROBERT JAMES;RING KELLEE GRIFFIN;DYAKONOV TATYANA;MIDDLEMISS DAVID
分类号 A61K31/40;A61K31/422;A61K31/426;A61K31/4439;A61K31/497;A61K31/506;A61P3/10;C07D207/16;C07D277/04;C07D401/12;C07D403/12;C07D413/12 主分类号 A61K31/40
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