发明名称 BENZOXAZINE AND QUINOXALINE DERIVATIVES AND USE THEREOF
摘要 FIELD: chemistry. ^ SUBSTANCE: described are compounds of formula ; or their pharmaceutically acceptable salts, where A is phenyl, X is CH2- or C=O; Y is O; k equals 1; m equals 0; R2 and R3 each independently represents hydrogen or alkyl, R4 is a group of formula or . Disclosed compounds have selective affinity to 5-HT6 and 5-HT2A receptors. Also described is a pharmaceutical composition containing said compounds and use of the said compounds in making a medicinal agent for treating diseased conditions of the central nervous system. ^ EFFECT: more effective treatment. ^ 49 cl, 1 tbl, 16 ex
申请公布号 RU2382036(C2) 申请公布日期 2010.02.20
申请号 RU20070110479 申请日期 2005.09.22
申请人 F.KHOFFMANN-LJA ROSH AG 发明人 BONKHAUS DUGLAS VILL'JAM;MARTIN RENE SHARON;SETKHOFER STIVEN;CHZHAN LI;CHZHAO SHU-KHAJ
分类号 A61K31/536;A61P25/00;C07D265/36;C07D413/04;C07D413/06 主分类号 A61K31/536
代理机构 代理人
主权项
地址