| 摘要 |
<p>(A) Cpds. of the general formula (I) R' = (1-4C)alkyl, (3-4C) alkenyl or (5-7C) cycloalkyl R2 = H, Me or Et X = H, F, Cl, Br, Me, MeS, MeO or CH3CO (B) Acid addn. salts of I. Oral and parenteral hypoglycaemics. Dose 100-500 mg/d. N-(2-methylaminoethyl)-p-methoxybenzene-sulphonamide (24.4 g.) was stirred with BrCN (10.6 g.) and 2N-NaOH (100 ml) at 20-30 deg., filtered, and recryst. from MeOH, giving the imidazoline, m.p. 104-7 deg.</p> |
