发明名称 |
NEW PYRROLE DERIVATIVE AS PHARMACEUTICAL AGENT |
摘要 |
PROBLEM TO BE SOLVED: To provide pyrazole derivatives as TGF-βsignal transduction inhibitors. SOLUTION: Provided are compounds having the structure of formula (I), wherein formulaαis a four, five, or six membered saturated ring; and X is C, O or S. COPYRIGHT: (C)2009,JPO&INPIT
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申请公布号 |
JP2009197016(A) |
申请公布日期 |
2009.09.03 |
申请号 |
JP20090108167 |
申请日期 |
2009.04.27 |
申请人 |
ELI LILLY & CO |
发明人 |
SAWYER JASON SCOTT;BEIGHT DOUGLAS W;CIAPETTI PAOLA;DECOLLO TODD VINCENT;ALEXANDER GLENN GODFREY;GOODSON THEODORE JR;HERRON DAVID KENT;LI HONG-YU;LIAO JUNKAI;MCMILLEN WILLIAM THOMAS;MILLER SHAWN CHRISTOPHER;MORT NICOLAS ANTHONY;YINGLING JONATHAN MICHAEL;SMITH EDWARD C R |
分类号 |
C07D471/04;A61K31/4162;A61K31/4439;A61K31/444;A61K31/4709;A61K31/496;A61K31/497;A61K31/501;A61K31/5383;A61K31/55;A61K45/00;A61P1/16;A61P3/10;A61P7/04;A61P9/10;A61P11/00;A61P13/12;A61P17/02;A61P17/12;A61P19/02;A61P21/00;A61P21/02;A61P25/28;A61P27/02;A61P29/00;A61P31/00;A61P31/18;A61P35/00;A61P37/02;A61P37/06;A61P37/08;A61P43/00;C07D401/12;C07D487/04;C07D498/04 |
主分类号 |
C07D471/04 |
代理机构 |
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代理人 |
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地址 |
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