发明名称 PYRROLOPYRAZINE KINASE INHIBITORS
摘要 The present invention relates to the use of novel pyrrolopyrazine derivatives of Formula (I), wherein the variables Q1 and R are defined as described herein, which inhibit JAK and SYK and are useful for the treatment of auto-immune and inflammatory diseases.
申请公布号 WO2009106445(A1) 申请公布日期 2009.09.03
申请号 WO2009EP51761 申请日期 2009.02.16
申请人 F. HOFFMANN-LA ROCHE AG;DU BOIS, DAISY, JOE;ELWORTHY, TODD, RICHARD;HENDRICKS, ROBERT, THAN;HERMANN, JOHANNES, CORNELIUS;KONDRU, RAMA, K.;LOU, YAN;OWENS, TIMOTHY, D.;PARK, JAEHYEON;SMITH, DAVID, BERNARD;SOTH, MICHAEL;YEE, CALVIN, WESLEY 发明人 DU BOIS, DAISY, JOE;ELWORTHY, TODD, RICHARD;HENDRICKS, ROBERT, THAN;HERMANN, JOHANNES, CORNELIUS;KONDRU, RAMA, K.;LOU, YAN;OWENS, TIMOTHY, D.;PARK, JAEHYEON;SMITH, DAVID, BERNARD;SOTH, MICHAEL;YEE, CALVIN, WESLEY
分类号 C07D487/04;A61K31/5025;A61P29/00;C07D519/00 主分类号 C07D487/04
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