发明名称 6,6-BICYCLIC RING SUBSTITUTED HETEROBICYCLIC PROTEIN KINASE INHIBITOR
摘要 PROBLEM TO BE SOLVED: To provide a compound inhibiting IGF-1R enzyme and useful for treatment and/or prevention of hyperproliferative diseases such as cancer, inflammation, psoriasis, allergy/asthma, disease and conditions of the immune system, disease and conditions of the central nervous system. SOLUTION: Compounds of formula (I) (wherein, X<SB>1</SB>, X<SB>2</SB>, X<SB>3</SB>, X<SB>4</SB>, X<SB>5</SB>, X<SB>6</SB>, X<SB>7</SB>, R<SP>1</SP>, and Q<SP>1</SP>are specifically defined) and pharmaceutically acceptable salts thereof, are provided. COPYRIGHT: (C)2009,JPO&INPIT
申请公布号 JP2009197013(A) 申请公布日期 2009.09.03
申请号 JP20090102856 申请日期 2009.04.21
申请人 OSI PHARMACEUTICALS INC 发明人 ARNOLD LEE D;CESARIO CARA;COATE HEATHER;CREW ANDREW PHILIP;DONG HANQING;FOREMAN KENNETH;HONDA AYAKO;LAUFER RADOSLAW;LI AN-HU;MULVIHILL KRISTEN MICHELLE;MULVIHILL MARK JOSEPH;NIGRO ANTHONY;PANICKER BIJOY;STEINIG ARNO G;SUN YINGCHUAN;WENG QINGHUA;WERNER DOUGLAS S;WYLE MICHAEL J;ZHANG TAO
分类号 C07D487/04;A61K31/437;A61K31/4985;A61K31/5025;A61K31/517;A61K31/519;A61K31/53;A61K31/5377;A61P7/02;A61P9/10;A61P11/06;A61P17/06;A61P29/00;A61P35/00;A61P37/06;A61P37/08;A61P43/00;C07D471/04 主分类号 C07D487/04
代理机构 代理人
主权项
地址